OX40

OX40

OX40 Overview

Molecule Name
Tumor necrosis factor receptor superfamily member 4
Synonyms
TNFRSF4,OX40,CD134,OX40L receptor,ACT35,TXGP1L
Drug Development Progress
Drugs in Clinical Trials27
Approved Drugs0
Highest Development StagePhase 3 Clinical
Target Synonym
ATC35 Antigen,OX40 Antigen,ACT35,IMD16,OX40,Receptors, OX40,ACT35 antigen,TNFRSF4,CD134,TNF Receptor Superfamily Member 4,TAX Transcriptionally-Activated Glycoprotein 1 Receptor,CD134 Antigen,TXGP1L,Tumor Necrosis Factor Receptor Superfamily, Member 4,Lymphoid Activation Antigene ACT35,OX40 Homologue,Tumor necrosis factor receptor superfamily member 4,Tax-Transcriptionally Activated Glycoprotein 1 Receptor,OX40 Cell Surface Antigen,OX40L receptor
Background
Tumor necrosis factor receptor superfamily member 4 (TNFRSF4) is also known as ACT35 antigen, OX40L receptor, TAX transcriptionally-activated glycoprotein 1 receptor, CD antigen CD134, OX40. OX40 / TNFRSF4 contains four TNFR-Cys repeats. TNFRSF4 is receptor for TNFSF4 / OX40L / GP34 and can interacts with TRAF2, TRAF3 and TRAF5.

OX40 Product List

Species
  • Human(5)
  • Cynomolgus / Rhesus macaque(3)
  • Mouse(3)
  • Rat(2)
  • Canine(1)
  • Rabbit(1)
Tag
  • Fc Tag(5)
  • His Tag(5)
  • His Tag & Avi Tag(3)
  • Fc Tag & Avi Tag(1)
  • Mouse IgG Fc Tag(1)
Host
  • HEK293(15)
Conjugate
  • Unconjugated(11)
  • Biotin-labeled(4)
Grade
  • RUO(15)
Low Endotoxin
  • Yes(4)
  • No(11)
MoleculeCat. No.Product NameSpeciesHostStructurePurityActivitySize&Price
OX40
HOTAvitag
OX0-C82E9
Biotinylated Cynomolgus / Rhesus macaque OX40 / TNFRSF4 / CD134 Protein, His,Avitag™ (MALS verified)
Cynomolgus / Rhesus macaque
HEK293
MALSSDS-PAGE
ELISA

$360.00

25ug
OX40
Human OX40 / TNFRSF4 / CD134 Protein, His Tag (Mass Spec & MALS verified)
Human
HEK293
MALSSDS-PAGE
ELISABLI

$405.00

100ug
OX40
Human OX40 / TNFRSF4 / CD134 Protein, Mouse IgG2a Fc Tag, low endotoxin (MALS verified)
Human
HEK293
MALSSDS-PAGE
ELISAFlow

$340.00

100ug
OX40
Human OX40 / TNFRSF4 / CD134 Protein, Fc Tag, low endotoxin (MALS verified)
Human
HEK293
MALSSDS-PAGE
ELISAFlow

$335.00

100ug
OX40
Biotinylated Human OX40 / TNFRSF4 / CD134 Protein, Avitag™,His Tag (MALS verified) (recommended for biopanning)
Human
HEK293
MALSSDS-PAGE
ELISABLI

$400.00

25ug
OX40
Cynomolgus / Rhesus macaque OX40 / TNFRSF4 / CD134 Protein, His Tag, low endotoxin (MALS verified)
Cynomolgus / Rhesus macaque
HEK293
MALSSDS-PAGE
ELISA

$360.00

100ug
OX40
Cynomolgus / Rhesus macaque OX40 / TNFRSF4 / CD134 Protein, Fc Tag (MALS verified)
Cynomolgus / Rhesus macaque
HEK293
MALSSDS-PAGE
ELISA

$275.00

100ug
OX40
Canine OX40 / TNFRSF4 / CD134 Protein, Fc Tag (MALS verified)
Canine
HEK293
MALSSDS-PAGE
ELISA

$360.00

100ug
OX40
Avitag
OX0-H82F7
Biotinylated Human OX40 Protein, Fc,Avitag™ (MALS verified)
Human
HEK293
MALSSDS-PAGE
ELISAFlow

$360.00

25ug
OX40
Mouse OX40 / TNFRSF4 / CD134 Protein, His Tag (MALS verified)
Mouse
HEK293
MALSSDS-PAGE
ELISA

$275.00

100ug
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Project NameProject StageMolecule TypeMolecule SourceDisease AreaIndication
OX40 mAb - 01LeadMonoclonalHumanized MouseAutoImmunityAutoimmune disease
Project Name
OX40 mAb - 01
Project Stage
Lead
Molecule Type
Monoclonal
Molecule Source
Humanized Mouse
Disease Area
AutoImmunity
Indication
Autoimmune disease
Resources

Clinical Drug Information

English NameResearch CodeHighest Development StageCompanyIndicationClinical Trial
RocatinlimabKHK-4083; AMG-451Phase 3 ClinicalAmgen Inc, Kyowa Hakko Kirin Co Ltd
Abdominal Pain; Asthma; Autoimmune Diseases; Colitis; Colitis, Ulcerative; Colonic Diseases; Dermatitis, Atopic; Digestive System Diseases; Gastrointestinal Diseases; Inflammatory Bowel Diseases; Intestinal Diseases; Prurigo Nodularis
Details
IvuxolimabPF-8600; PF-04518600Phase 3 ClinicalPfizer Inc
Bone metastases; Breast Neoplasms; Carcinoma; Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Leukemia, Myeloid, Acute; Lymphoma, Follicular; Neoplasms; Ovarian Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Solid tumours; Triple Negative Breast Neoplasms
Details
INBRX-106INBRX-106; ES-102; ES102Phase 3 ClinicalInhibrx
Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Carcinoma, Transitional Cell; Head and Neck Neoplasms; Melanoma; Neoplasms; Solid tumours; Squamous Cell Carcinoma of Head and Neck; Stomach Neoplasms
Details
GSK3174998GSK3174998; GSK 3174998; GSK-3174998Phase 2 ClinicalGlaxosmithkline Plc
Multiple Myeloma; Neoplasms
Details
TelazorlimabGBR-830; ISB-830Phase 2 ClinicalGlenmark Pharmaceuticals Ltd
Dermatitis, Atopic
Details
TavolimabMEDI-0562Phase 2 ClinicalMedimmune
Carcinoma, Ovarian Epithelial; Carcinoma, Squamous Cell; Fallopian Tube Neoplasms; Head and Neck Neoplasms; Melanoma; Neoplasms, Squamous Cell; Ovarian Neoplasms; Peritoneal Neoplasms; Solid tumours; Squamous Cell Carcinoma of Head and Neck
Details
HX-111HX-111; HX111Phase 2 ClinicalHanx Biopharmaceuticals (Wuhan) Co Ltd
Hematologic Neoplasms; Lymphoma; Solid tumours
Details
CS-01CS01; CS-01Phase 2 ClinicalZhongshan Constimulus Bio Co Ltd
Solid tumours
Details
BrivekimigSAR-442970; SAR442970Phase 2 ClinicalSanofi
Colitis, Ulcerative; Crohn Disease; Diabetes Mellitus, Type 1; Glomerulonephritis; Glomerulosclerosis, Focal Segmental; Hidradenitis Suppurativa; Inflammation; Nephrosis
Details
IMG-007IMG-007Phase 2 Clinical
Alopecia Areata; Dermatitis, Atopic; Eczema
Details
BAT-6026BAT-6026Phase 2 ClinicalBio-Thera Solutions Ltd, Sunshine GuoJian Pharmaceutical (Shanghai) Co Ltd
Autoimmune Diseases; Dermatitis, Atopic; Solid tumours
Details
GimistotugBGB-A445Phase 2 ClinicalBeOne Medicines Ltd
Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Carcinoma, Transitional Cell; Melanoma; Nasopharyngeal Carcinoma; Solid tumours; Squamous Cell Carcinoma of Head and Neck
Details
Recombinant human anti-OX40 monoclonal antibody (Livzon Group)Phase 1 ClinicalLivzon Pharmaceutical Group Inc
Neoplasms
Details
SL-279252TAK-252; SL-279252Phase 1 ClinicalShattuck Labs Inc, Takeda Pharmaceutical Co Ltd
Adenocarcinoma; Astrocytoma; Carcinoma, Basosquamous; Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Carcinoma, Squamous Cell; Carcinoma, Transitional Cell; Esophageal Neoplasms; Gastroesophageal Junction Neoplasms; Hodgkin Disease; Lymphoma, Large B-Cell, Diffuse; Melanoma; Solid tumours; Squamous Cell Carcinoma of Head and Neck; Stomach Neoplasms
Details
FS-120FS-120Phase 1 ClinicalF-Star
Neoplasm Metastasis; Neoplasms
Details
CudarolimabIBI-101Phase 1 Clinical
Neoplasms; Solid tumours
Details
RevdofilimabABBV-368; PR-1628103Phase 1 ClinicalAbbvie Inc
Carcinoma, Non-Small-Cell Lung; Head and Neck Neoplasms; Neoplasms; Solid tumours; Triple Negative Breast Neoplasms
Details
SHR-1806SHR-1806Phase 1 ClinicalJiangsu Hengrui Medicine Co Ltd, Suzhou Suncadia Biopharmaceuticals Co Ltd
Neoplasms
Details
BMS-986178BMS-986178Phase 1 ClinicalBristol-Myers Squibb Company
Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma, B-Cell; Lymphoma, B-Cell, Marginal Zone; Lymphoma, Follicular; Lymphoma, Mantle-Cell; Neoplasms; Solid tumours; Waldenstrom Macroglobulinemia
Details
EMB-09EMB-09Phase 1 ClinicalShanghai Epimab Biotherapeutics, Inc
Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Colorectal Neoplasms; Endometrial Neoplasms; Hepatitis B, Chronic; Melanoma; Nasopharyngeal Carcinoma; Neoplasms; Ovarian Neoplasms; Small Cell Lung Carcinoma; Solid tumours; Squamous Cell Carcinoma of Head and Neck; Stomach Neoplasms; Triple Negative Breast Neoplasms
Details
PeptiCRAd-1Valo-D102; PeptiCRAd-1Phase 1 ClinicalValor Biotherapeutics
Carcinoma, Non-Small-Cell Lung; Colorectal Neoplasms; Liposarcoma, Myxoid; Neoplasms; Osteosarcoma; Sarcoma; Sarcoma, Synovial; Skin Melanoma; Triple Negative Breast Neoplasms
Details
CenzestotugYH-002Phase 1 Clinical
Solid tumours
Details
SAR-446422SAR446422; SAR-446422Phase 1 ClinicalSanofi
Autoimmune Diseases
Details
STAR-0310ISB-830-X8; STAR-0310; STR-310Phase 1 ClinicalIchnos Sciences Inc
Dermatitis, Atopic
Details
HFB-3010HFB-301001; HFB-3010Phase 1 ClinicalHiFiBiO Therapeutics
Carcinoma, Hepatocellular; Carcinoma, Renal Cell; Melanoma; Sarcoma; Solid tumours; Squamous Cell Carcinoma of Head and Neck; Uterine Neoplasms
Details
HLX-51HLX-51Phase 1 Clinical
Lymphoma; Solid tumours
Details
MEDI-6469MEDI-6469; AGX-051Phase 1 ClinicalAgonOx Inc, Astrazeneca Plc, Providence Cancer Center, Providence Health & Services
Colorectal Neoplasms; Head and Neck Neoplasms; Liver Neoplasms; Lung Neoplasms; Lymphoma; Melanoma; Metastatic breast cancer; Neoplasms; Prostatic Neoplasms; Solid tumours
Details
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