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CCR5

CCR5 Overview

English NameC-C chemokine receptor type 5Approved Drugs1
Drugs in Clinical Trials13Target SynonymCCR-5,Chemokine (C-C Motif) Receptor 5 (Gene/Pseudogene),C-C Motif Chemokine Receptor 5 A159A,Chemokine Recptor CCR5 Delta32,C-C Chemokine Receptor Type 5,Chemokine Receptor CCR5,CD195 Antigen,C-C CKR-5,CCCKR5,IDDM22,CKR-5,CKR5,Receptors, CCR5,C-C Motif Chemokine Receptor 5,CD195,CHEMR13,CCR5,HIV-1 fusion coreceptor,C-C Motif Chemokine Receptor 5 (Gene/Pseudogene),Chemokine (C-C Motif) Receptor 5,CC-CKR-5,CMKBR5
Highest Development StageApproved
English NameC-C chemokine receptor type 5
Target SynonymCCR-5,Chemokine (C-C Motif) Receptor 5 (Gene/Pseudogene),C-C Motif Chemokine Receptor 5 A159A,Chemokine Recptor CCR5 Delta32,C-C Chemokine Receptor Type 5,Chemokine Receptor CCR5,CD195 Antigen,C-C CKR-5,CCCKR5,IDDM22,CKR-5,CKR5,Receptors, CCR5,C-C Motif Chemokine Receptor 5,CD195,CHEMR13,CCR5,HIV-1 fusion coreceptor,C-C Motif Chemokine Receptor 5 (Gene/Pseudogene),Chemokine (C-C Motif) Receptor 5,CC-CKR-5,CMKBR5
Approved Drugs1
Drugs in Clinical Trials13
Highest Development StageApproved

CCR5 Product List

  • Product Category

    Protein (4)Cell (1)

  • Product Status

    Launched (5)

  • Species

    Human (4)Mouse (1)

  • Tag

    His Tag & Flag Tag (2)- (2)GFP Tag (1)

  • Conjugate

    Unconjugated (3)- (1)GFP Fusion (1)

CCR5 Synonyms

CCR5,CMKBR5,CD195,CC-CKR-5,CHEMR13

Clinical Drug Information

English NameResearch CodeHighest Development StageCompanyIndicationClinical Trial
Cenicriviroc mesylateCCR5/CCR2 antagonist; TBR-652; CVC; TAK-652Phase 3 ClinicalTakeda Pharmaceutical Co Ltd, Tobira Therapeutics IncAIDS Dementia Complex; Cholangitis, Sclerosing; Cognition Disorders; Coronavirus Disease 2019 (COVID-19); Diabetes Mellitus, Type 2; Hepatic Insufficiency; HIV Infections; Liver Cirrhosis; Metabolic Dysfunction-Associated Steatotic Liver Disease; Obesity; Prediabetic State
Details
SB-728-TSB-728mR-T; SB-728-TPhase 2 ClinicalSangamo BiosciencesHIV Infections
Details
VicrivirocSCH-D; MK-4176; SCH-417; Sch-417690Phase 2 ClinicalMerck & Co IncAcquired Immunodeficiency Syndrome; Colorectal Neoplasms; HIV Infections
Details
LeronlimabPA-14; PRO-140; HuPRO-140Phase 2 ClinicalProgenics Pharmaceuticals IncColorectal Neoplasms; Coronavirus Disease 2019 (COVID-19); Graft vs Host Disease; HIV Infections; Metabolic Dysfunction-Associated Steatotic Liver Disease; Rectal Neoplasms; Solid tumours; Triple Negative Breast Neoplasms
Details
BMS-813160BMS-813160Phase 2 ClinicalBristol-Myers Squibb CompanyAdenocarcinoma; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Pancreatic Ductal; Colorectal Neoplasms; Diabetic Nephropathies; Hyperplasia; Pancreatic Neoplasms
Details
RAP-103RAP-160; RAP-701; RAP-164; RAP-310; RAP-163; RAP-103Phase 2 ClinicalRapid PharmaceuticalsAlzheimer Disease; Hepatitis B; Neuralgia; Ovarian Neoplasms; Prostatic Neoplasms; Psoriasis
Details
Cenicriviroc mesylate/TropifexorLJC-242Phase 2 ClinicalNovartis Pharma AgMetabolic Dysfunction-Associated Steatotic Liver Disease
Details
AGT 103-TAGT 103-TPhase 1 ClinicalAmerican Gene Technologies International IncHIV Infections
Details
ThioravirocPhase 1 ClinicalShanghai Institute Of Materia Medica, Chinese Academy Of SciencesAmyotrophic Lateral Sclerosis; HIV Infections; Multiple Sclerosis
Details
BMS-687681BMS-687681Phase 1 ClinicalBristol-Myers Squibb CompanyNeoplasms
Details
SB-728-HSCSB-728-HSC; SB-728-HSPC; SB-728mR-HSPCPhase 1 ClinicalSangamo BiosciencesHIV Infections
Details
vMIP (Guangzhou Hongrun Biotech)Phase 1 ClinicalGuangzhou Hongrun Biotechnology Co LtdPneumonia
Details
LF-0376LF-0376Phase 1 ClinicalWuxi Hillhouse biomedicine Technology Co LtdColorectal Neoplasms; Liver Neoplasms; Lymphoma; Lymphoma, Large B-Cell, Diffuse; Pancreatic Neoplasms; Solid tumours
Details

Marketed Drug Information

English NameResearch CodeHighest Development StageCompanyEarliest Brand NameEarliest Approval CountryEarliest IndicationEarliest Approval CompanyEarliest Approval DateIndicationClinical Trial
MaravirocMVC; UK-427857ApprovedViiv HealthcareCelsentri, SelzentryUnited StatesHIV InfectionsViiv Healthcare Co2007-08-06Acquired Immunodeficiency Syndrome; Acute Lung Injury; AIDS Dementia Complex; Arthritis, Rheumatoid; Cardiovascular Diseases; Cognition Disorders; Coronavirus Disease 2019 (COVID-19); HIV Infections; Hypertriglyceridemia; Inflammation; Ischemic Stroke; Kidney Diseases; Primary Graft Dysfunction; Rejection of lung transplantation; Sarcoma, Kaposi; Stroke
Details
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